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1、防己的藥理作用及臨床應(yīng)用研究進(jìn)展 [摘要]防己,又名粉防己、漢防己,是我國傳統(tǒng)常用中藥之一,味苦、辛,性寒,具有祛風(fēng)濕、止痹痛、利水消腫等功效,中醫(yī)主要用于治療風(fēng)濕痹證、水腫、小便不利、腳氣腫痛、濕瘡腫毒等。防己的主要成分為雙芐基異喹啉類生物堿,包括粉防己堿、防己諾林堿等,現(xiàn)代藥理學(xué)研究發(fā)現(xiàn)防己及其主要成分在抗炎、抗病原微生物、抗腫瘤、抗高血壓、抗心律失常、抗心肌缺血、抗纖維化、抗矽肺、抑制瘢痕等方面均具有廣泛的藥理活性,應(yīng)用前景廣闊。臨床上常將防己與其他中藥組方配伍應(yīng)用,主要用于治療類風(fēng)濕關(guān)節(jié)炎、心血管疾病、腫瘤、高血壓、肝腹水
2、等疾病,取得較好療效;常用的代表方劑有防己茯苓湯、防己黃芪湯、己椒藶黃丸、宣痹湯、復(fù)方漢防己顆粒等。該文對防己的藥理作用及臨床應(yīng)用進(jìn)行了綜述,為中藥防己的進(jìn)一步開發(fā)利用提供參考?! 關(guān)鍵詞]防己;藥理作用;臨床應(yīng)用;類風(fēng)濕關(guān)節(jié)炎;心血管疾病;腫瘤 [Abstract]StephaniaTetrandraeRadixisoneofthecommontraditionalChinesemedicines,whichhasbitterandpungenttasteaswellascoldproperties.Itcansubsidee
3、dema,getridofrheumatismandrelievepain.Therefore,itismainlyusedforthetreatmentofrheumatismarthralgia,edema,dysuria,athlete'sfoot,swollenwetsoresandotherdiseasesintraditionalChinesemedicine(TCM).StephaniaTetrandraeRadixismainlycomposedofdual-benzylisoquinolinealkaloids,i
4、ncludingtetrandrine,fangchinolineandsoon.ModernpharmacologyresearchshowsthatStephaniaTetrandraeRadixanditsmaincomponentshaveawiderangeofpharmacologicalactivitiesintheanti-inflammatory,anti-pathogenicmicroorganisms,anti-tumor,anti-hypertensive,anti-arrhythmic,anti-myoca
5、rdialischemia,anti-fibrosis,anti-silicosis,inhibitingscarandotheraspects,withbroadapplicationprospect.StephaniaTetrandraeRadixisoftenappliedwithcompatibilityofotherChinesemedicinesinclinically,andhasachievedobviouseffectsinthetreatmentofrheumatoidarthritis,cardiovascul
6、ardisease,cancer,hypertension,liverascitesandotherdiseases.Therearesomerepresentativeprescriptions,suchasFangjiFulingdecoction,F(xiàn)angjihuangqidecoction,JijiaoLizhuangpill,Xuanbidecoction,andcompoundHanfangjigranule.Inthispaper,thepharmacologicaleffectsandclinicalapplicat
7、ionsofStephaniaTetrandraeRadixinthepasttenyearswerereviewed,providingreferenceforitsfurtherdevelopmentandapplication. [Keywords]StephaniaTetrandraeRadix;pharmacologicaleffects;clinicalapplication;rheumatismarthralgia;anti-inflammatory;rheumatoidarthritis;cardiovascula
8、rdisease;tumor 防己,又名粉防己、?h防己,是傳統(tǒng)的常用中藥之一,始載于《神農(nóng)本草經(jīng)》,一直被作為祛風(fēng)濕藥使用。防己自古以來分為漢防己和木防己兩大類,一般習(xí)慣所稱的漢防己實(shí)際上是防己科的粉防己,而不是馬兜鈴科的漢中防己